Synthesis of 1,2-cis-Homoiminosugars Derived from GlcNAc and GalNAc Exploiting a β-Amino Alcohol Skeletal Rearrangement Y Blériot, N Auberger, Y Jagadeesh, C Gauthier, G Prencipe, AT Tran, ... Organic letters 16 (21), 5512-5515, 2014 | 36 | 2014 |
DDQ-Promoted Benzylic/Allylic sp3 C–H Activation for the Stereoselective Intramolecular C–N Bond Formation: Applications to the Total Synthesis of (−)-Codonopsinine, (+)-5 … M Lingamurthy, Y Jagadeesh, K Ramakrishna, BV Rao The Journal of Organic Chemistry 81 (4), 1367-1377, 2016 | 28 | 2016 |
Synthesis of 1,2-trans-2-Acetamido-2-deoxyhomoiminosugars Y Blériot, AT Tran, G Prencipe, Y Jagadeesh, N Auberger, S Zhu, ... Organic Letters 16 (21), 5516-5519, 2014 | 25 | 2014 |
Total synthesis of (−)-codonopsinol and (+)-2-epi codonopsinol via acid catalyzed amido cyclisation Y Jagadeesh, JS Reddy, BV Rao, JL Swarnalatha Tetrahedron 66 (6), 1202-1207, 2010 | 25 | 2010 |
Efficacy assessment of an uncharged reactivator of nop-inhibited acetylcholinesterase based on tetrahydroacridine pyridine-aldoxime hybrid in mouse compared to pralidoxime AG Calas, AS Hanak, N Jaffré, A Nervo, J Dias, C Rousseau, ... Biomolecules 10 (6), 858, 2020 | 17 | 2020 |
Total synthesis of radicamine B and 5-epi-radicamine B Y Jagadeesh, BV Rao Tetrahedron letters 52 (48), 6366-6369, 2011 | 16 | 2011 |
The synthesis of (1S, 8aS)-1-hydroxyindolizidine using a stereoselective Grignard addition to an N-benzyl-3-deoxy sugar imine derived from D-Glucose Y Jagadeesh, B Chandrasekhar, BV Rao Tetrahedron: Asymmetry 21 (18), 2314-2318, 2010 | 15 | 2010 |
Chiron approach to (−)-deoxocuscohygrine Y Jagadeesh, KKS Reddy, BV Rao Tetrahedron: Asymmetry 22 (14-15), 1485-1489, 2011 | 11 | 2011 |
Synthesis of pyrrolidine-based analogues of 2-acetamidosugars as N-acetyl-d-glucosaminidase inhibitors AT Tran, B Luo, Y Jagadeesh, N Auberger, J Désiré, S Nakagawa, A Kato, ... Carbohydrate research 409, 56-62, 2015 | 9 | 2015 |
A common synthetic approach for seven and eight-membered polyhydroxylated iminocyclitols Y Jagadeesh, K Ramakrishna, BV Rao Tetrahedron: Asymmetry 23 (9), 697-702, 2012 | 9 | 2012 |
Iminosugar C‐Glycosides Work as Pharmacological Chaperones of NAGLU, a Glycosidase Involved in MPS IIIB Rare Disease** S Zhu, Y Jagadeesh, AT Tran, S Imaeda, A Boraston, DS Alonzi, ... Chemistry–A European Journal 27 (44), 11291-11297, 2021 | 7 | 2021 |
Chemoselective Hydrogenation of 6‐Alkynyl‐3‐fluoro‐2‐pyridinaldoximes: Access to First‐in‐Class 6‐Alkyl‐3‐Fluoro‐2‐pyridinaldoxime Scaffolds as New Reactivators of Sarin … J Yerri, J Dias, MR Nimmakayala, F Razafindrainibe, C Courageux, ... Chemistry–A European Journal 26 (65), 15035-15044, 2020 | 7 | 2020 |
γ-Aminoalcohol rearrangement applied to pentahydroxylated azepanes provides pyrrolidines epimeric to homoDMDP Y Jagadeesh, AT Tran, B Luo, N Auberger, J Désiré, S Nakagawa, A Kato, ... Organic & Biomolecular Chemistry 13 (11), 3446-3456, 2015 | 5 | 2015 |
Sonogashira Reaction of Bromofluoropyridinaldoxime Nuclei: Convergent Synthesis of Functionalized 2‐and 3‐Fluoropyridine Scaffolds J Yerri, R Baati European Journal of Organic Chemistry 2018 (30), 4161-4165, 2018 | 4 | 2018 |
Sonogashira Cross‐Coupling Reaction of Bromocyanofluoro Pyridine Compounds: Access to 5‐and 6‐Alkynylfluoropyridinamidoximes Scaffolds F Razafindrainibe, C Voros, Y Jagadeesh, NM Reddy, A Tissier, K Mardy, ... European Journal of Organic Chemistry 2021 (30), 4393-4397, 2021 | 2 | 2021 |
Cycloaddition of Benzyne with Alkoxy-Substituted Pyrroline-N-oxides: Unexpected Rearrangement to an N-Phenylpyrrole FM Cordero, BB Khairnar, A Ranzenigo, A Brandi SynOpen 2 (01), 0025-0029, 2018 | 2 | 2018 |
Divergent Synthesis of Various 2-Aryl Iminocyclitols from (R)-p-Hydroxyphenylglycine VK Jain Synthesis 51 (24), 4635-4644, 2019 | 1 | 2019 |
Influence of A1,3 Strain on the Stereochemical Outcome of Acid‐Mediated Amido Cyclization in the Synthesis of 2‐(4‐Methoxyphenyl)‐3,4‐(dihydroxy)piperidines K Ramakrishna, Y Jagadeesh, KVS Ramakrishna, JL Rao, BV Rao European Journal of Organic Chemistry 2016 (9), 1693-1701, 2016 | 1 | 2016 |
Hydroxy-pyridinaldoxime scaffolds R Baati, R Brown, D José, A Maryan-instone, F Nachon, J Yerri, C Voros US Patent App. 18/043,958, 2024 | | 2024 |
6-Substituted 3-Fluoro-2-Pyridinaldoxime, 3-Fluoro-2-pyridine hydroxamic acid, and 3-Fluoro-2-Pyridinamidoxime scaffolds R Baati, J Yerri, D José US Patent 11,370,772, 2022 | | 2022 |