Raphael Labruere
Raphael Labruere
Associate prof. of Bioorganic Chemistry, Univ. Paris-Saclay
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Self‐Immolative Spacers: Kinetic Aspects, Structure–Property Relationships, and Applications
A Alouane, R Labručre, T Le Saux, F Schmidt, L Jullien
Angewandte Chemie International Edition 54 (26), 7492-7509, 2015
“Self‐Immolative” Spacer for Uncaging with Fluorescence Reporting
R Labručre, A Alouane, T Le Saux, I Aujard, P Pelupessy, A Gautier, ...
Angewandte Chemie International Edition 51 (37), 9344-9347, 2012
Biochemical and structural analysis of the binding determinants of a vascular endothelial growth factor receptor peptidic antagonist
B Gautier, V Goncalves, D Diana, R Di Stasi, F Teillet, C Lenoir, ...
Journal of medicinal chemistry 53 (11), 4428-4440, 2010
Anti–Methicillin-Resistant Staphylococcus aureus Nanoantibiotics
R Labručre, AJ Sona, E Turos
Frontiers in Pharmacology 10, 2019
Selbstzerlegende Spacer: kinetische Aspekte, Struktur‐Eigenschafts‐Beziehungen und Anwendungen
A Alouane, R Labručre, T Le Saux, F Schmidt, L Jullien
Angewandte Chemie 127 (26), 7600-7619, 2015
Design, Synthesis, and Biological Evaluation of the First Podophyllotoxin Analogues as Potential Vascular‐Disrupting Agents
R Labručre, B Gautier, M Testud, J Seguin, C Lenoir, S Desbčne‐Finck, ...
ChemMedChem 5 (12), 2016-2025, 2010
Light Activation for the Versatile and Accurate Kinetic Analysis of Disassembly of Self‐Immolative Spacers
A Alouane, R Labručre, T Le Saux, I Aujard, S Dubruille, F Schmidt, ...
Chemistry-A European Journal 19 (35), 11717-11724, 2013
Anticancer boron-containing prodrugs responsive to oxidative stress from the tumor microenvironment
H Maslah, C Skarbek, S Pethe, R Labručre
European Journal of Medicinal Chemistry 207, 112670, 2020
Design and Effective Synthesis of the First 4-Aza-2, 3-didehydropodophyllotoxin Rigid Aminologue: AN-Methyl-4-[(3, 4, 5-trimethoxyphenyl) amino)]-1, 2-dihydroquinoline-lactone
R Labručre, P Helissey, S Desbčne-Finck, S Giorgi-Renault
The Journal of organic chemistry 73 (9), 3642-3645, 2008
Polyamine-based analogs and conjugates as antikinetoplastid agents
E Jagu, S Pomel, S Pethe, PM Loiseau, R Labručre
European Journal of Medicinal Chemistry 139, 982-1015, 2017
Poly (vinyl benzoate) nanoparticles for molecular delivery: Studies on their preparation and in vitro properties
R Labručre, R Sicard, R Cormier, E Turos, L West
Journal of Controlled Release 148 (2), 234-240, 2010
Arylboronate prodrugs of doxorubicin as promising chemotherapy for pancreatic cancer
C Skarbek, S Serra, H Maslah, E Rascol, R Labručre
Bioorganic chemistry 91, 103158, 2019
Design, synthesis and in vitro antikinetoplastid evaluation of N-acylated putrescine, spermidine and spermine derivatives
E Jagu, R Djilali, S Pomel, F Ramiandrasoa, S Pethe, R Labručre, ...
Bioorganic & medicinal chemistry letters 25 (2), 207-209, 2015
Disassembly Kinetics of Quinone‐Methide‐Based Self‐Immolative Spacers that Contain Aromatic Nitrogen Heterocycles
A Alouane, R Labručre, KJ Silvestre, T Le Saux, F Schmidt, L Jullien
Chemistry–An Asian Journal 9 (5), 1334-1340, 2014
Synthesis and in vitro antikinetoplastid activity of polyamine–hydroxybenzotriazole conjugates
E Jagu, S Pomel, A Diez-Martinez, F Ramiandrasoa, RL Krauth-Siegel, ...
Bioorganic & medicinal chemistry 25 (1), 84-90, 2017
Synthesis and antikinetoplastid evaluation of bis (benzyl) spermidine derivatives
E Jagu, S Pomel, A Diez-Martinez, E Rascol, S Pethe, PM Loiseau, ...
European journal of medicinal chemistry 150, 655-666, 2018
In‐Cell Generation of Anticancer Phenanthridine Through Bioorthogonal Cyclization in Antitumor Prodrug Development
H Maslah, C Skarbek, C Gourson, MA Plamont, S Pethe, L Jullien, ...
Angewandte Chemie 133 (45), 24245-24249, 2021
Spermine-NBD as fluorescent probe for studies of the polyamine transport system in Leishmania donovani
E Jagu, S Pomel, S Pethe, JC Cintrat, PM Loiseau, R Labručre
Bioorganic & medicinal chemistry letters 29 (14), 1710-1713, 2019
A chemically encoded timer for dual molecular delivery at tailored ranges and concentrations
S Serra, A Alouane, T Le Saux, S Huvelle, R Plasson, F Schmidt, L Jullien, ...
Chemical Communications 54 (49), 6396-6399, 2018
Attenuating the size and molecular carrier capabilities of polyacrylate nanoparticles by a hydrophobic fluorine effect
R Labručre, E Turos
Bioorganic & medicinal chemistry 20 (16), 5042-5045, 2012
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