| SLC-0111 enaminone analogs, 3/4-(3-aryl-3-oxopropenyl) aminobenzenesulfonamides, as novel selective subnanomolar inhibitors of the tumor-associated carbonic anhydrase isoform IX WM Eldehna, MF Abo-Ashour, E Berrino, D Vullo, HA Ghabbour, ... Bioorganic chemistry 83, 549-558, 2019 | 57 | 2019 |
| Rho-kinase inhibitors in the management of glaucoma E Berrino, CT Supuran Expert Opinion on Therapeutic Patents 29 (10), 817-827, 2019 | 45 | 2019 |
| Synthesis and Evaluation of Carbonic Anhydrase Inhibitors with Carbon Monoxide Releasing Properties for the Management of Rheumatoid Arthritis E Berrino, L Milazzo, L Micheli, D Vullo, A Angeli, M Bozdag, A Nocentini, ... Journal of medicinal chemistry 62 (15), 7233-7249, 2019 | 40 | 2019 |
| Novel approaches for designing drugs that interfere with pH regulation E Berrino, CT Supuran Expert opinion on drug discovery 14 (3), 231-248, 2019 | 37 | 2019 |
| Azidothymidine (AZT)“clicked” into 1, 2, 3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual Hybrid Inhibitors E Berrino, A Angeli, DD Zhdanov, AP Kiryukhina, A Milaneschi, A De Luca, ... Journal of Medicinal Chemistry, 2020 | 32 | 2020 |
| Synthesis and carbonic anhydrase inhibitory properties of novel 4-(2-aminoethyl) benzenesulfonamide-dipeptide conjugates H Küçükbay, N Buğday, FZ Küçükbay, E Berrino, G Bartolucci, S Del Prete, ... Bioorganic chemistry 83, 414-423, 2019 | 29 | 2019 |
| Novel sulfamide-containing compounds as selective carbonic anhydrase I inhibitors E Berrino, S Bua, M Mori, M Botta, VS Murthy, V Vijayakumar, Y Tamboli, ... Molecules 22 (7), 1049, 2017 | 28 | 2017 |
| Advances in microwave-assisted synthesis and the impact of novel drug discovery E Berrino, CT Supuran Expert opinion on drug discovery 13 (9), 861-873, 2018 | 23 | 2018 |
| New thiopyrimidine-benzenesulfonamide conjugates as selective carbonic anhydrase II inhibitors: synthesis, in vitro biological evaluation, and molecular docking studies HT Abdel-Mohsen, AM El Kerdawy, MA Omar, E Berrino, AS Abdelsamie, ... Bioorganic & Medicinal Chemistry 28 (5), 115329, 2020 | 22 | 2020 |
| 4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors S Salerno, E Barresi, G Amendola, E Berrino, C Milite, AM Marini, ... Journal of medicinal chemistry 61 (13), 5765-5770, 2018 | 19 | 2018 |
| New sulfonamides containing organometallic-acylhydrazones: synthesis, characterisation and biological evaluation as inhibitors of human carbonic anhydrases Y Huentupil, L Peña, N Novoa, E Berrino, R Arancibia, CT Supuran Journal of Enzyme Inhibition and Medicinal Chemistry 34 (1), 451-458, 2019 | 18 | 2019 |
| Inhibition of α-, β-, γ-, and δ-carbonic anhydrases from bacteria and diatoms with N′-aryl-N-hydroxy-ureas E Berrino, M Bozdag, S Del Prete, FAS Alasmary, LS Alqahtani, ... Journal of enzyme inhibition and medicinal chemistry 33 (1), 1194-1198, 2018 | 18 | 2018 |
| Synthesis of novel benzenesulfamide derivatives with inhibitory activity against human cytosolic carbonic anhydrase I and II and Vibrio cholerae α- and β-class … S Bua, E Berrino, S Del Prete, VS Murthy, V Vijayakumar, Y Tamboli, ... Journal of enzyme inhibition and medicinal chemistry 33 (1), 1125-1136, 2018 | 16 | 2018 |
| 1, 2, 4-Trisubstituted imidazolinones with dual carbonic anhydrase and p38 mitogen-activated protein kinase inhibitory activity HH Georgey, FM Manhi, WR Mahmoud, NA Mohamed, E Berrino, ... Bioorganic chemistry 82, 109-116, 2019 | 13 | 2019 |
| Bioorganometallic derivatives of 4-hydrazino-benzenesulphonamide as carbonic anhydrase inhibitors: synthesis, characterisation and biological evaluation J Brichet, R Arancibia, E Berrino, CT Supuran Journal of Enzyme Inhibition and Medicinal Chemistry 35 (1), 622-628, 2020 | 11 | 2020 |
| A class of carbonic anhydrase IX/XII–selective carboxylate inhibitors RA Alhameed, E Berrino, Z Almarhoon, A El-Faham, CT Supuran Journal of Enzyme Inhibition and Medicinal Chemistry 35 (1), 549-554, 2020 | 10 | 2020 |
| N-aryl-N’-ureido-O-sulfamates as potent and selective inhibitors of hCA VB over hCA VA: deciphering the binding mode of new potential agents in mitochondrial dysfunctions G Poli, M Bozdag, E Berrino, A Angeli, T Tuccinardi, F Carta, CT Supuran Bioorganic Chemistry, 103896, 2020 | 9 | 2020 |
| Carbonic anhydrase inhibitors for the treatment of epilepsy and obesity E Berrino, F Carta Carbonic Anhydrases, 311-329, 2019 | 9 | 2019 |
| Carbonic Anhydrase Inhibitors of Different Structures Dilate Pre-Contracted Porcine Retinal Arteries T Eysteinsson, H Gudmundsdottir, AO Hardarson, E Berrino, S Selleri, ... International Journal of Molecular Sciences 20 (3), 467, 2019 | 9 | 2019 |
| In silico identification and biological evaluation of antioxidant food components endowed with IX and XII hCA inhibition G Costa, A Maruca, R Rocca, FA Ambrosio, E Berrino, F Carta, F Mesiti, ... Antioxidants 9 (9), 775, 2020 | 7* | 2020 |
