Extrapyramidal side effects of antipsychotics are linked to their association kinetics at dopamine D2 receptors DA Sykes, H Moore, L Stott, N Holliday, JA Javitch, JR Lane, SJ Charlton Nature communications 8 (1), 763, 2017 | 192 | 2017 |
Unravelling intrinsic efficacy and ligand bias at G protein coupled receptors: A practical guide to assessing functional data LA Stott, DA Hall, ND Holliday Biochemical pharmacology 101, 1-12, 2016 | 44 | 2016 |
Potent and selective N-(4-sulfamoylphenyl) thiourea-based GPR55 agonists S Yrjölä, T Parkkari, D Navia-Paldanius, T Laitinen, AA Kaczor, T Kokkola, ... European journal of medicinal chemistry 107, 119-132, 2016 | 25 | 2016 |
Extrapyramidal side effects of antipsychotics are linked to their association kinetics at dopamine D2 receptors. Nat Commun. 2017; 8 (1): 763 DA Sykes, H Moore, L Stott, N Holliday, JA Javitch, JR Lane, SJ Charlton Epub 2017/10/04. https://doi. org/10.1038/s41467-017-00716-z PMID: 28970469, 0 | 5 | |
The identification of GPR52 agonist HTL0041178, a potential therapy for schizophrenia and related psychiatric disorders S Poulter, N Austin, R Armstrong, M Barnes, SJ Bucknell, A Higueruelo, ... ACS Medicinal Chemistry Letters 14 (4), 499-505, 2023 | 4 | 2023 |
Characterisation of inverse agonism of the orphan-G protein-coupled receptor GPR52 by cannabinoid ligands Cannabidiol and O-1918 LA Stott, CA Brighton, J Brown, R Mould, KA Bennett, R Newman, ... Heliyon 7 (6), 2021 | 4 | 2021 |
Effect of HTL0045725, a selective agonist of the orphan receptor GPR52, on kinase and transcription factor phosphorylation in striatal neurons E Sergeev, L Stott, SJ Bradley, KA Bennett, AJH Brown, SP Watson, ... Neuroscience Applied 1, 100412, 2022 | 2 | 2022 |
The neutrophil dynamic mass redistribution assay as a medium throughput primary cell screening assay LA Stott, AD la Rochelle, S Brown, G Osborne, CJ Hutchings, S Poulter, ... Journal of Pharmacology and Experimental Therapeutics 389 (1), 19-31, 2024 | 1 | 2024 |
Validation of a label-free assay to determine chemokine responses in primary human neutrophils L Stott, G Osborne, K Bennett, S Poulter, C Hutchings, M Barnes BRITISH JOURNAL OF PHARMACOLOGY 177 (11), 2509-2511, 2020 | | 2020 |
Comparison of radioligand and TR-FRET binding techniques at the histamine H-4 receptor D Tippett, LA Stott, G Osborne, M Barnes BRITISH JOURNAL OF PHARMACOLOGY 176 (16), 2988-2989, 2019 | | 2019 |
Determination of agonist intrinsic efficacies at the dopamine D2 receptor LA Stott University of Nottingham, 2017 | | 2017 |
Comparison of Radioligand and TR-FRET Binding Techniques at the Histamine H DN Tippett, LA Stott, G Osborne, M Barnes membranes 4, 4, 0 | | |