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Marinella Roberti
Marinella Roberti
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Synthesis and biological evaluation of resveratrol and analogues as apoptosis-inducing agents
M Roberti, D Pizzirani, D Simoni, R Rondanin, R Baruchello, C Bonora, ...
Journal of medicinal chemistry 46 (16), 3546-3554, 2003
3012003
Pterostilbene and 3′-hydroxypterostilbene are effective apoptosis-inducing agents in MDR and BCR-ABL-expressing leukemia cells
M Tolomeo, S Grimaudo, A Di Cristina, M Roberti, D Pizzirani, M Meli, ...
The international journal of biochemistry & cell biology 37 (8), 1709-1726, 2005
2032005
Heterocyclic and phenyl double-bond-locked combretastatin analogues possessing potent apoptosis-inducing activity in HL60 and in MDR cell lines
D Simoni, G Grisolia, G Giannini, M Roberti, R Rondanin, L Piccagli, ...
Journal of medicinal chemistry 48 (3), 723-736, 2005
1952005
Multitarget drug design strategy: quinone–tacrine hybrids designed to block amyloid-β aggregation and to exert anticholinesterase and antioxidant effects
E Nepovimova, E Uliassi, J Korabecny, LE Pena-Altamira, S Samez, ...
Journal of medicinal chemistry 57 (20), 8576-8589, 2014
1822014
Galloflavin (CAS 568‐80‐9): a novel inhibitor of lactate dehydrogenase
M Manerba, M Vettraino, L Fiume, G Di Stefano, A Sartini, E Giacomini, ...
ChemMedChem 7 (2), 311-317, 2012
1762012
Non-ATP competitive protein kinase inhibitors
L Garuti, M Roberti, G Bottegoni
Current medicinal chemistry 17 (25), 2804-2821, 2010
1622010
Irreversible protein kinase inhibitors
L Garuti, M Roberti, G Bottegoni
Current medicinal chemistry 18 (20), 2981-2994, 2011
1412011
Tetramethylguanidine (TMG)-catalyzed addition of dialkyl phosphites to α, β-unsaturated carbonyl compounds, alkenenitriles, aldehydes, ketones and imines
D Simoni, FP Invidiata, M Manferdini, I Lampronti, R Rondanin, M Roberti, ...
Tetrahedron letters 39 (41), 7615-7618, 1998
1391998
Galloflavin, a new lactate dehydrogenase inhibitor, induces the death of human breast cancer cells with different glycolytic attitude by affecting distinct signaling pathways
F Farabegoli, M Vettraino, M Manerba, L Fiume, M Roberti, G Di Stefano
European Journal of Pharmaceutical Sciences 47 (4), 729-738, 2012
1372012
Strong bicyclic guanidine base-promoted Wittig and Horner− Wadsworth− Emmons reactions
D Simoni, M Rossi, R Rondanin, A Mazzali, R Baruchello, C Malagutti, ...
Organic letters 2 (24), 3765-3768, 2000
1332000
Berberine and its metabolites: relationship between physicochemical properties and plasma levels after administration to human subjects
S Spinozzi, C Colliva, C Camborata, M Roberti, C Ianni, F Neri, ...
Journal of Natural Products 77 (4), 766-772, 2014
1322014
Synthesis and antiproliferative activity of some benzimidazole-4, 7-dione derivatives
L Garuti, M Roberti, M Malagoli, T Rossi, M Castelli
Bioorganic & medicinal chemistry letters 10 (19), 2193-2195, 2000
1262000
Heterocycle-containing retinoids. Discovery of a novel isoxazole arotinoid possessing potent apoptotic activity in multidrug and drug-induced apoptosis-resistant cells
D Simoni, M Roberti, FP Invidiata, R Rondanin, R Baruchello, C Malagutti, ...
Journal of medicinal chemistry 44 (14), 2308-2318, 2001
1152001
Tacrine-resveratrol fused hybrids as multi-target-directed ligands against Alzheimer's disease
J Jeřábek, E Uliassi, L Guidotti, J Korábečný, O Soukup, V Sepsova, ...
European Journal of Medicinal Chemistry 127, 250-262, 2017
1122017
Nitrogen-containing heterocyclic quinones: a class of potential selective antitumor agents.
L Garuti, M Roberti, D Pizzirani
Mini Reviews in Medicinal Chemistry 7 (5), 481-489, 2007
1052007
Synthesis and antiviral activity of some N-benzenesulphonylbenzimidazoles
L Garuti, M Roberti, C Cermelli
Bioorganic & medicinal chemistry letters 9 (17), 2525-2530, 1999
1051999
Antioxidant activity of hydroxystilbene derivatives in homogeneous solution
R Amorati, M Lucarini, V Mugnaini, GF Pedulli, M Roberti, D Pizzirani
The Journal of organic chemistry 69 (21), 7101-7107, 2004
1032004
Identification of biphenyl-based hybrid molecules able to decrease the intracellular level of Bcl-2 protein in Bcl-2 overexpressing leukemia cells
D Pizzirani, M Roberti, S Grimaudo, A Di Cristina, RM Pipitone, ...
Journal of medicinal chemistry 52 (21), 6936-6940, 2009
1022009
Identification of a Terphenyl Derivative that Blocks the Cell Cycle in the G0−G1 Phase and Induces Differentiation in Leukemia Cells
M Roberti, D Pizzirani, M Recanatini, D Simoni, S Grimaudo, D Cristina, ...
Journal of medicinal chemistry 49 (10), 3012-3018, 2006
1022006
Stilbene-based anticancer agents: resveratrol analogues active toward HL60 leukemic cells with a non-specific phase mechanism
D Simoni, M Roberti, FP Invidiata, E Aiello, S Aiello, P Marchetti, ...
Bioorganic & Medicinal Chemistry Letters 16 (12), 3245-3248, 2006
992006
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