89Zr-Immuno-Positron Emission Tomography in Oncology: State-of-the-Art 89Zr Radiochemistry S Heskamp, R Raavé, O Boerman, M Rijpkema, V Goncalves, F Denat Bioconjugate Chemistry 28 (9), 2211-2223, 2017 | 169 | 2017 |
A fluorescence-based assay for N-myristoyltransferase activity V Goncalves, JA Brannigan, E Thinon, TO Olaleye, R Serwa, S Lanzarone, ... Analytical Biochemistry 421 (1), 342-344, 2012 | 87 | 2012 |
Discovery of Plasmodium vivax N-Myristoyltransferase Inhibitors: Screening, Synthesis, and Structural Characterization of their Binding Mode V Goncalves, JA Brannigan, D Whalley, KH Ansell, B Saxty, AA Holder, ... Journal of Medicinal Chemistry 55 (7), 3578-3582, 2012 | 74 | 2012 |
Structure-Based Design of Potent and Selective Leishmania N-Myristoyltransferase Inhibitors JA Hutton, V Goncalves, JA Brannigan, D Paape, MH Wright, TM Waugh, ... Journal of medicinal chemistry 57 (20), 8664-8670, 2014 | 72 | 2014 |
Direct comparison of the in vitro and in vivo stability of DFO, DFO* and DFOcyclo* for 89Zr-immunoPET R Raavé, G Sandker, P Adumeau, CB Jacobsen, F Mangin, M Meyer, ... European Journal of Nuclear Medicine and Molecular Imaging 46, 1966-1977, 2019 | 68 | 2019 |
On-resin cyclization of peptide ligands of the vascular endothelial growth factor receptor 1 by copper (I)-catalyzed 1, 3-dipolar azide–alkyne cycloaddition V Goncalves, B Gautier, A Regazzetti, P Coric, S Bouaziz, C Garbay, ... Bioorganic & medicinal chemistry letters 17 (20), 5590-5594, 2007 | 61 | 2007 |
(R)-NODAGA-PSMA: a versatile precursor for radiometal labeling and nuclear imaging of PSMA-positive tumors E Gourni, C Canovas, V Goncalves, F Denat, PT Meyer, HR Maecke PLoS One 10 (12), e0145755, 2015 | 56 | 2015 |
Site‐Specific Dual Labeling of Proteins on Cysteine Residues with Chlorotetrazines C Canovas, M Moreau, C Bernhard, A Oudot, M Guillemin, F Denat, ... Angewandte Chemie International Edition 57 (33), 10646-10650, 2018 | 50 | 2018 |
Development of a chemiluminescent screening assay for detection of vascular endothelial growth factor receptor 1 ligands. V Goncalves, B Gautier, C Garbay, M Vidal, N Inguimbert Analytical biochemistry 366 (1), 108-110, 2007 | 49 | 2007 |
Targeting the Proangiogenic VEGF-VEGFR Protein-Protein Interface with Drug-like Compounds by In Silico and In Vitro Screening. B Gautier, MA Miteva, V Goncalves, F Huguenot, P Coric, S Bouaziz, ... Chemistry & biology 18 (12), 1631, 2011 | 47 | 2011 |
Towards the elaboration of new gold-based optical theranostics PE Doulain, R Decréau, C Racoeur, V Goncalves, L Dubrez, A Bettaieb, ... Dalton Transactions 44, 4874-4883, 2015 | 43 | 2015 |
Biochemical and structural analysis of the binding determinants of a vascular endothelial growth factor receptor peptidic antagonist B Gautier, V Goncalves, D Diana, R Di Stasi, F Teillet, C Lenoir, ... Journal of medicinal chemistry 53 (11), 4428-4440, 2010 | 43 | 2010 |
Rational design, structure, and biological evaluation of cyclic peptides mimicking the vascular endothelial growth factor V Goncalves, B Gautier, P Coric, S Bouaziz, C Lenoir, C Garbay, M Vidal, ... Journal of medicinal chemistry 50 (21), 5135-5146, 2007 | 41 | 2007 |
DMAP‐BODIPY Alkynes: A Convenient Tool for Labeling Biomolecules for Bimodal PET–Optical Imaging B Brizet, V Goncalves, C Bernhard, PD Harvey, F Denat, C Goze Chemistry–A European Journal 20 (40), 12933-12944, 2014 | 34 | 2014 |
Site-specific near-infrared fluorescent labelling of proteins on cysteine residues with meso-chloro-substituted heptamethine cyanine dyes C Canovas, PS Bellaye, M Moreau, A Romieu, F Denat, V Goncalves Organic & Biomolecular Chemistry 16 (45), 8831-8836, 2018 | 33 | 2018 |
BODIPY: a highly versatile platform for the design of bimodal imaging probes D Lhenry, M Larrouy, C Bernhard, V Goncalves, O Raguin, P Provent, ... Chemistry–A European Journal 21 (37), 13091-13099, 2015 | 27 | 2015 |
Design of bimodal ligands of neurotensin receptor 1 for positron emission tomography imaging and fluorescence-guided surgery of pancreatic cancer E Renard, PA Dancer, C Portal, F Denat, A Prignon, V Goncalves Journal of Medicinal Chemistry 63 (5), 2426-2433, 2019 | 23 | 2019 |
Structure‐based design of a bicyclic peptide antagonist of the vascular endothelial growth factor receptors V Goncalves, B Gautier, C Garbay, M Vidal, N Inguimbert Journal of peptide science: an official publication of the European Peptide …, 2008 | 21 | 2008 |
Modular Assembly of Multimodal Imaging Agents through an Inverse Electron Demand Diels–Alder Reaction C Canovas, M Moreau, JM Vrigneaud, PS Bellaye, B Collin, F Denat, ... Bioconjugate Chemistry 30 (3), 888-897, 2019 | 20 | 2019 |
Direct subphthalocyanine conjugation to bombesin vs. indirect conjugation to its lipidic nanocarrier Y Bernhard, E Gigot, V Goncalves, M Moreau, N Sok, P Richard, ... Organic & Biomolecular Chemistry 14 (19), 4511-4518, 2016 | 16 | 2016 |