A fluorescence-based assay for N-myristoyltransferase activity V Goncalves, JA Brannigan, E Thinon, TO Olaleye, R Serwa, S Lanzarone, ... Analytical Biochemistry 421 (1), 342-344, 2012 | 61 | 2012 |
Discovery of Plasmodium vivax N-Myristoyltransferase Inhibitors: Screening, Synthesis, and Structural Characterization of their Binding Mode V Goncalves, JA Brannigan, D Whalley, KH Ansell, B Saxty, AA Holder, ... Journal of Medicinal Chemistry 55 (7), 3578-3582, 2012 | 55 | 2012 |
On-resin cyclization of peptide ligands of the Vascular Endothelial Growth Factor Receptor 1 by copper (I)-catalyzed 1, 3-dipolar azide-alkyne cycloaddition V Goncalves, B Gautier, A Regazzetti, P Coric, S Bouaziz, C Garbay, ... Bioorganic & medicinal chemistry letters 17 (20), 5590-5594, 2007 | 53 | 2007 |
Structure-Based Design of Potent and Selective Leishmania N-Myristoyltransferase Inhibitors JA Hutton, V Goncalves, JA Brannigan, D Paape, MH Wright, TM Waugh, ... Journal of medicinal chemistry 57 (20), 8664-8670, 2014 | 49 | 2014 |
Targeting the Proangiogenic VEGF-VEGFR Protein-Protein Interface with Drug-like Compounds by In Silico and In Vitro Screening. B Gautier, MA Miteva, V Goncalves, F Huguenot, P Coric, S Bouaziz, ... Chemistry & biology 18 (12), 1631, 2011 | 42 | 2011 |
Development of a chemiluminescent screening assay for detection of vascular endothelial growth factor receptor 1 ligands. V Goncalves, B Gautier, C Garbay, M Vidal, N Inguimbert Analytical biochemistry 366 (1), 108-110, 2007 | 41 | 2007 |
Rational design, structure, and biological evaluation of cyclic peptides mimicking the vascular endothelial growth factor V Goncalves, B Gautier, P Coric, S Bouaziz, C Lenoir, C Garbay, M Vidal, ... Journal of medicinal chemistry 50 (21), 5135-5146, 2007 | 37 | 2007 |
Biochemical and structural analysis of the binding determinants of a vascular endothelial growth factor receptor peptidic antagonist B Gautier, V Goncalves, D Diana, R Di Stasi, F Teillet, C Lenoir, ... Journal of medicinal chemistry 53 (11), 4428-4440, 2010 | 36 | 2010 |
89Zr-Immuno-Positron Emission Tomography in Oncology: State-of-the-Art 89Zr Radiochemistry S Heskamp, R Raavé, O Boerman, M Rijpkema, V Goncalves, F Denat Bioconjugate chemistry 28 (9), 2211-2223, 2017 | 35 | 2017 |
(R)-NODAGA-PSMA: A Versatile Precursor for Radiometal Labeling and Nuclear Imaging of PSMA-Positive Tumors E Gourni, C Canovas, V Goncalves, F Denat, PT Meyer, HR Maecke PloS one 10 (12), e0145755, 2015 | 29 | 2015 |
Towards the elaboration of new gold-based optical theranostics PE Doulain, R Decréau, C Racoeur, V Goncalves, L Dubrez, A Bettaieb, ... Dalton Transactions 44, 4874-4883, 2015 | 28 | 2015 |
DMAP‐BODIPY Alkynes: A Convenient Tool for Labeling Biomolecules for Bimodal PET–Optical Imaging B Brizet, V Goncalves, C Bernhard, PD Harvey, F Denat, C Goze Chemistry-A European Journal 20 (40), 12933-12944, 2014 | 24 | 2014 |
BODIPY: A Highly Versatile Platform for the Design of Bimodal Imaging Probes D Lhenry, M Larrouy, C Bernhard, V Goncalves, O Raguin, P Provent, ... Chemistry-A European Journal 21 (37), 13091-13099, 2015 | 18 | 2015 |
Structure‐based design of a bicyclic peptide antagonist of the vascular endothelial growth factor receptors V Goncalves, B Gautier, C Garbay, M Vidal, N Inguimbert Journal of peptide science: an official publication of the European Peptide …, 2008 | 17 | 2008 |
Site‐Specific Dual Labeling of Proteins on Cysteine Residues with Chlorotetrazines C Canovas, M Moreau, C Bernhard, A Oudot, M Guillemin, F Denat, ... Angewandte Chemie International Edition 57 (33), 10646-10650, 2018 | 12 | 2018 |
MA‐NOTMP: A Triazacyclononane Trimethylphosphinate Based Bifunctional Chelator for Gallium Radiolabelling of Biomolecules S Poty, P Désogère, J Šimeček, C Bernhard, V Goncalves, C Goze, ... ChemMedChem 10 (9), 1475-1479, 2015 | 9 | 2015 |
Total chemical synthesis of the D2 domain of human VEGF receptor 1 V Goncalves, B Gautier, F Huguenot, P Leproux, C Garbay, M Vidal, ... Journal of peptide science: an official publication of the European Peptide …, 2009 | 9 | 2009 |
Direct subphthalocyanine conjugation to bombesin vs. indirect conjugation to its lipidic nanocarrier Y Bernhard, E Gigot, V Goncalves, M Moreau, N Sok, P Richard, ... Organic & Biomolecular Chemistry 14 (19), 4511-4518, 2016 | 8 | 2016 |
Structure-guided optimization of quinoline inhibitors of Plasmodium N-myristoyltransferase V Goncalves, JA Brannigan, A Laporte, AS Bell, SM Roberts, AJ Wilkinson, ... MedChemComm 8 (1), 191-197, 2017 | 5 | 2017 |
Peptides as antagonists of the VEGF receptors V Goncalves, B Gautier, C Lenoir, C Garbay, M Vidal, N Inguimbert Pharmachem, 15-19, 2006 | 5 | 2006 |